MK-5 with vented cover (polycarbonate 

To Order Contact us: stephen@expresspharmapulse.com

MK-3903

B2431-5
EUR 414

MK-886

B2517-5
EUR 175

MK 886

B6684-5 5 mg
EUR 137

MK-0941

B1207-5
EUR 185

MK-8931

B1315-5
EUR 512

MK-5108

B1344-5
EUR 262

MK 571

B7023-5 5 mg
EUR 128
Description: MK 571 (L-660,711) is a novel potent and selective antagonist of leukotriene D4 receptor with Ki values of 0.22 nM and 2.1 nM in guinea pig and human lung membranes, respectively [1].

MK-4101

B7803-5 5 mg
EUR 261
Description: IC50: 1.5 ?mol/L for in mouse Light II cells by Gli_luc assayMK-4101 is a Hedgehog (Hh) signaling pathway inhibitor.Abnormal activation of the Hedgehog (Hh) signaling pathway is reported in the pathogenesis of various cancers, such as medulloblastoma and basal cell carcinoma.

MK-4827

9462-5
EUR 305

MK-3102

9599-5
EUR 457

MK 0893

A3608-5 5 mg
EUR 415
Description: MK 0893 is an inhibitor of both glucagon receptor and IGF-1R with IC50 values of 6.6nM and 6nM, respectively [1, 2].

MK-0591

A3609-5 5 mg
EUR 284
Description: MK-0591, an analog of MK-886 is a potent and orally active leukotriene biosynthesis inhibitor with an IC50 value of 600 ng/ml.

MK-0812

A3611-5 5 mg
EUR 379
Description: MK-0812 is an antagonist of chemokine receptor CCR-2 [1].C-C chemokine receptor type 2 (CCR-2) is a chemokine receptor expressing on monocytes and macrophages and plays a critical and apparently non-redundant role in orchestrating the trafficking of monocytes to tissues [1].

MK-0974

A3612-5 5 mg
EUR 395
Description: MK-0974 (Telcagepant) is a highly potent, selective, and orally bioavailable antagonist of CGRP receptor with IC50 value of 0.77 nM [1].

MK-2894

A3613-5 5 mg
EUR 357
Description: MK-2894 is a highly potent and selective inhibitor of EP4 receptor with IC50 value of 2.5 nM [1].

MK-3207

A3615-5 5 mg
EUR 340
Description: MK-3207 is a new, highly selective CGRP receptor antagonist that is approximately 40- to 65-fold more potent than telcagepant for the human CGRP receptor. The IC50 is 0.12 nM and The Ki value is 0.024 nM. It is highly selective versus human AM1, AM2, CTR, and AMY3.

MK-4827

A3617-5 5 mg
EUR 209
Description: MK-4827 is a novel, selective and orally bioavailable PARP1/PARP2 inhibitor with IC50 of 3.8 nM and 2.1 nM, respevctively.MK-4827 has shown great activity against cancer cells with mutant BRCA-1 and BRCA-2; >330-fold selective against PARP3, V-PARP and Tank1 [1].

MK-5172

A3618-5 5 mg
EUR 154
Description: MK-5172 is a selective inhibitor of Hepatitis C Virus NS3/4a Protease [1].Hepatitis C (HCV) virus is a member of the Flaviviridae family of viruses in the Hepacivirus genus and encoded by a 9.6-kb positive strand RNA genome [2].

MK-6892

A3623-5 5 mg
EUR 502
Description: Description:IC50 Value: 4.0 nM (Ki for Human GPR109A) [1]MK-6892 is a highly potential GPR109A agonists.in vitro: . Despite the increased serum shift of these compounds, the representative 1e was highly potent

MK-8033

A3624-5 5 mg
EUR 466
Description: MK-8033 is a c-MET inhibitor in clinical trials. MK8033 is a selective small-molecule inhibitor, ATP competitive. Phase I investigation of the cMet inhibitor MK-8033 is ongoing.

MK-0752

A4006-5 5 mg
EUR 247
Description: MK-0752 is a potent gamma secretase inhibitor in clinical development (IC50 ~50 nM).

MK-2048

A4072-5 5 mg
EUR 270
Description: MK-2048 is a second generation inhibitor of HIV-1 integrase with IC50 values of 0.075 ?M and 0.08 ?M for subtype B and subtype C integrase, respectively.Integration of viral cDNA into the host genome is one of the definitive features of retrovirus replication.

MK-5 with vented cover (polycarbonate